865273-97-8
865273-97-8 structure
- Name: ERAP1-IN-1
- Chemical Name: ERAP1-IN-1
- CAS Number: 865273-97-8
- Molecular Formula: C20H21F3N2O5S
- Molecular Weight: 458.45
- Catalog: Research Areas Inflammation/Immunology
- Create Date: 2020-01-23 22:03:51
- Modify Date: 2024-01-11 16:30:09
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ERAP1-IN-1 is an endoplasmic reticulum aminopeptidase 1 (ERAP1) inhibitor. ERAP1-IN-1 competitively inhibits ERAP1 activity towards a nonamer peptide representative of physiological substrates[1].
| Name | ERAP1-IN-1 |
|---|
| Description | ERAP1-IN-1 is an endoplasmic reticulum aminopeptidase 1 (ERAP1) inhibitor. ERAP1-IN-1 competitively inhibits ERAP1 activity towards a nonamer peptide representative of physiological substrates[1]. |
|---|---|
| Related Catalog | |
| Target |
ERAP1[1] |
| In Vitro | ERAP1-IN-1 allosterically activates ERAP1’s hydrolysis of fluorogenic and chromogenic amino acid substratesv[1]. ERAP1-IN-1 (50 µM) exhibits specific inhibition of ERAP1 in the cellular context[1]. |
| References |
| Molecular Formula | C20H21F3N2O5S |
|---|---|
| Molecular Weight | 458.45 |
| Hazard Codes | Xi |
|---|