Name | PI3KC2α-IN-2 |
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Description | PI3KC2α-IN-2 is a potent and selective PI3KC2α inhibitor (IC50: 121 nM). PI3KC2α-IN-2 interacts with the ATP-binding site of PI3KC2α.. PI3KC2α-IN-2 can be used in the research of thrombosis, diabetes and cancers[1]. |
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Related Catalog | |
Target |
PI3KC2α:121 nM (IC50) PI3KC2β:1399 nM (IC50) PI3KC2γ:>10 μM (IC50) |
In Vitro | PI3KC2α-IN-2 (PITCOIN2) is selective against PI3KC2γ but showed micromolar activity on PI3KC2β[1]. |
Molecular Formula | C25H20N6O3S2 |
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Molecular Weight | 516.59 |