Name | PKCiota-IN-1 |
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Description | PKCiota-IN-1 (compound 51) is a potent PKCiota (PKC-ι) inhibitor with an IC50 of 2.7 nM. PKCiota-IN-1 also inhibits PKC-α and PKC-ε with IC50s of 45 nM and 450 nM, respectively[1]. |
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Related Catalog | |
Target |
PKCι:2.7 nM (IC50) PKCα:45 nM (IC50) PKCε:450 nM (IC50) |
References |
Molecular Formula | C25H22FN5O |
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Molecular Weight | 427.47 |