FSHR agonist 1
Modify Date: 2024-04-06 22:04:47
FSHR agonist 1 structure
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Common Name | FSHR agonist 1 | ||
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| CAS Number | 1256776-89-2 | Molecular Weight | 467.62 | |
| Density | N/A | Boiling Point | N/A | |
| Molecular Formula | C26H33N3O3S | Melting Point | N/A | |
| MSDS | N/A | Flash Point | N/A | |
Use of FSHR agonist 1FSHR agonist 1 is a high affinity and allosteric follicle stimulating hormone receptor (FSHR) agonist with a pEC50 of 7.72. FSHR agonist 1 formes extensive interactions with the TMD to directly activate FSHR[1]. |
| Name | FSHR agonist 1 |
|---|
| Description | FSHR agonist 1 is a high affinity and allosteric follicle stimulating hormone receptor (FSHR) agonist with a pEC50 of 7.72. FSHR agonist 1 formes extensive interactions with the TMD to directly activate FSHR[1]. |
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| Related Catalog | |
| Target |
pEC50: 7.72 (FSHR)[1] |
| In Vitro | FSHR agonist 1 (compound 21f) 与 FSHR TMD 口袋的结合诱导 TM6 和 TM7 向内运动，这直接导致 FSHR 激活[1]。 FSHR agonist 1 (compound 21f) 可以高效激活 FSHR、LHCGR 和 TSHR，而对 FSHR 的激活效力比 LHCGR（pEC50 为 6.26）和 TSHR（pEC50 为 6.48）高 10 倍以上[1]。 |
| References |
| Molecular Formula | C26H33N3O3S |
|---|---|
| Molecular Weight | 467.62 |