Endomorphin 2 TFA

Modify Date: 2024-01-12 15:54:10

Endomorphin 2 TFA Structure
Endomorphin 2 TFA structure
Common Name Endomorphin 2 TFA
CAS Number 1276124-00-5 Molecular Weight 685.69
Density N/A Boiling Point N/A
Molecular Formula C34H38F3N5O7 Melting Point N/A
MSDS N/A Flash Point N/A

 Use of Endomorphin 2 TFA


Endomorphin 2 TFA, a high affinity, highly selective agonist of the μ-opioid receptor, displays reasonable affinities for kappa3 binding sites, with Ki value between 20 and 30 nM[1].

 Names

Name Endomorphin 2 TFA

 Endomorphin 2 TFA Biological Activity

Description Endomorphin 2 TFA, a high affinity, highly selective agonist of the μ-opioid receptor, displays reasonable affinities for kappa3 binding sites, with Ki value between 20 and 30 nM[1].
Related Catalog
Target

Ki: 20-30 nM (kappa3 opioid receptor)[1]

References

[1]. Goldberg IE, et al. Pharmacological characterization of endomorphin-1 and endomorphin-2 in mouse brain. J Pharmacol Exp Ther. 1998 Aug;286(2):1007-13.

 Chemical & Physical Properties

Molecular Formula C34H38F3N5O7
Molecular Weight 685.69
Storage condition 2-8℃