1276124-00-5

1276124-00-5 structure

Name: Endomorphin 2 TFA
Chemical Name: Endomorphin 2 TFA
CAS Number: 1276124-00-5
Molecular Formula: C₃₄H₃₈F₃N₅O₇
Molecular Weight: 685.69
Catalog: Signaling Pathways GPCR/G Protein Opioid Receptor
Create Date: 2019-06-01 15:58:33
Modify Date: 2024-01-12 15:54:10
Endomorphin 2 TFA, a high affinity, highly selective agonist of the μ-opioid receptor, displays reasonable affinities for kappa3 binding sites, with Ki value between 20 and 30 nM[1].

Name	Endomorphin 2 TFA

Description	Endomorphin 2 TFA, a high affinity, highly selective agonist of the μ-opioid receptor, displays reasonable affinities for kappa3 binding sites, with Ki value between 20 and 30 nM[1].
Related Catalog	Signaling Pathways >> GPCR/G Protein >> Opioid Receptor Signaling Pathways >> Neuronal Signaling >> Opioid Receptor Research Areas >> Neurological Disease
Target	Ki: 20-30 nM (kappa3 opioid receptor)[1]
References	[1]. Goldberg IE, et al. Pharmacological characterization of endomorphin-1 and endomorphin-2 in mouse brain. J Pharmacol Exp Ther. 1998 Aug;286(2):1007-13.