DC-CPin711

Modify Date: 2024-01-10 18:46:02

DC-CPin711 Structure
DC-CPin711 structure
Common Name DC-CPin711
CAS Number 2447559-21-7 Molecular Weight 386.45
Density N/A Boiling Point N/A
Molecular Formula C23H22N4O2 Melting Point N/A
MSDS N/A Flash Point N/A

 Use of DC-CPin711


DC-CPin711 is a potent and selective inhibitor of CREB-binding protein (CBP) bromodomain with an IC50 of 0.0626 μM. DC-CPin711 arrests cell cycle at G1 phase and induces apoptosis[1].

 Names

Name DC-CPin711

 DC-CPin711 Biological Activity

Description DC-CPin711 is a potent and selective inhibitor of CREB-binding protein (CBP) bromodomain with an IC50 of 0.0626 μM. DC-CPin711 arrests cell cycle at G1 phase and induces apoptosis[1].
Related Catalog
Target

IC50: 0.0626 μM (CBP bromodomain)[1]

References

[1]. Chen Y, et al. Design, synthesis, and biological evaluation of tetrahydroquinolin derivatives as potent inhibitors of CBP bromodomain. Bioorg Chem. 2020 Aug;101:103991.

 Chemical & Physical Properties

Molecular Formula C23H22N4O2
Molecular Weight 386.45