2447559-21-7

2447559-21-7 structure

2447559-21-7 structure

Name: DC-CPin711
Chemical Name: DC-CPin711
CAS Number: 2447559-21-7
Molecular Formula: C₂₃H₂₂N₄O₂
Molecular Weight: 386.45
Catalog: Signaling Pathways Apoptosis Apoptosis
Create Date: 2022-09-01 19:28:27
Modify Date: 2024-01-10 18:46:02
DC-CPin711 is a potent and selective inhibitor of CREB-binding protein (CBP) bromodomain with an IC50 of 0.0626 μM. DC-CPin711 arrests cell cycle at G1 phase and induces apoptosis[1].

Name	DC-CPin711

Description	DC-CPin711 is a potent and selective inhibitor of CREB-binding protein (CBP) bromodomain with an IC50 of 0.0626 μM. DC-CPin711 arrests cell cycle at G1 phase and induces apoptosis[1].
Related Catalog	Signaling Pathways >> Apoptosis >> Apoptosis Research Areas >> Cancer Signaling Pathways >> Epigenetics >> Epigenetic Reader Domain
Target	IC50: 0.0626 μM (CBP bromodomain)[1]
References	[1]. Chen Y, et al. Design, synthesis, and biological evaluation of tetrahydroquinolin derivatives as potent inhibitors of CBP bromodomain. Bioorg Chem. 2020 Aug;101:103991.

Molecular Formula	C₂₃H₂₂N₄O₂
Molecular Weight	386.45