CB1R Allosteric modulator 3
Modify Date: 2024-07-23 18:48:28
CB1R Allosteric modulator 3 structure
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Common Name | CB1R Allosteric modulator 3 | ||
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| CAS Number | 2633686-36-7 | Molecular Weight | 376.84 | |
| Density | N/A | Boiling Point | N/A | |
| Molecular Formula | C22H17ClN2O2 | Melting Point | N/A | |
| MSDS | N/A | Flash Point | N/A | |
Use of CB1R Allosteric modulator 3CB1R Allosteric modulator 3, a novel analogs derived from the 2-phenylindole scaffold, is a CB1R positive allosteric modulator. CB1R Allosteric modulator 3 has potent inhibition of cAMP and β-Arrestin with EC50 values of 0.018 μM and 1.241 μM[1]. |
| Name | CB1R Allosteric modulator 3 |
|---|
| Description | CB1R Allosteric modulator 3, a novel analogs derived from the 2-phenylindole scaffold, is a CB1R positive allosteric modulator. CB1R Allosteric modulator 3 has potent inhibition of cAMP and β-Arrestin with EC50 values of 0.018 μM and 1.241 μM[1]. |
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| Related Catalog | |
| Target |
CB1 |
| In Vitro | CB1R Allosteric modulator 3 has potent inhibition of cAMP and β-Arrestin with EC50 values of 0.018 μM and 1.241 μM. CB1R Allosteric modulator 3 can enhance CB1R ago-PAM activity because of small lipophilic functional groups on the ortho-position of the GAT211 site-III phenyl ring[1]. |
| References |
| Molecular Formula | C22H17ClN2O2 |
|---|---|
| Molecular Weight | 376.84 |