MRS 1754

Modify Date: 2024-01-08 07:34:18

MRS 1754 Structure
MRS 1754 structure
Common Name MRS 1754
CAS Number 264622-58-4 Molecular Weight 486.52200
Density 1.38g/cm3 Boiling Point N/A
Molecular Formula C26H26N6O4 Melting Point N/A
MSDS Chinese USA Flash Point N/A

 Use of MRS 1754


MRS 1754 is a selective antagonist radioligand for A2B adenosine receptor with very low affinity for A1 and A3 receptors of both humans and rats[1].

 Names

Name N-(4-cyanophenyl)-2-[4-(2,6-dioxo-1,3-dipropyl-7H-purin-8-yl)phenoxy]acetamide
Synonym More Synonyms

 MRS 1754 Biological Activity

Description MRS 1754 is a selective antagonist radioligand for A2B adenosine receptor with very low affinity for A1 and A3 receptors of both humans and rats[1].
Related Catalog
Target

A2B Adenosine Receptor[1]

In Vitro The most potent displacer of [3H]MRS 1754 binding is MRS 1754. The Ki value for displacement of [3H]MRS 1754 binding to human A2B receptors expressed in HEK-293 cell membranes is 1.45±0.21 nM[1].
References

[1]. Ji X, et al. [3H]MRS 1754, a selective antagonist radioligand for A(2B) adenosine receptors. Biochem Pharmacol. 2001 Mar 15;61(6):657-63.

 Chemical & Physical Properties

Density 1.38g/cm3
Molecular Formula C26H26N6O4
Molecular Weight 486.52200
Exact Mass 486.20200
PSA 134.80000
LogP 3.33548
Storage condition 2-8℃

 Safety Information

Safety Phrases 22-24/25

 Synonyms

MRS 1754 hydrate
MRS 1754
ML 9 hydrochloride
Lopac-M-6316
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