CYP3A4-IN-1

Modify Date: 2024-09-13 07:53:02

CYP3A4-IN-1 Structure
CYP3A4-IN-1 structure
Common Name CYP3A4-IN-1
CAS Number 2771297-34-6 Molecular Weight 559.72
Density N/A Boiling Point N/A
Molecular Formula C31H37N5O3S Melting Point N/A
MSDS N/A Flash Point N/A

 Use of CYP3A4-IN-1


CYP3A4-IN-1 (compound 5a) is a potent cytochrome P450 3A4 (CYP3A4) inhibitor with an IC50 value of 0.085 µM[1].

 Names

Name CYP3A4-IN-1

 CYP3A4-IN-1 Biological Activity

Description CYP3A4-IN-1 (compound 5a) is a potent cytochrome P450 3A4 (CYP3A4) inhibitor with an IC50 value of 0.085 µM[1].
Related Catalog
Target

CYP3A4:0.085 μM (IC50)

References

[1]. Samuels ER, et al. An increase in side-group hydrophobicity largely improves the potency of ritonavir-like inhibitors of CYP3A4. Bioorg Med Chem. 2020 Mar 15;28(6):115349.

 Chemical & Physical Properties

Molecular Formula C31H37N5O3S
Molecular Weight 559.72