Xanthine amine congener

Modify Date: 2024-01-07 19:52:47

Xanthine amine congener Structure
Xanthine amine congener structure
Common Name Xanthine amine congener
CAS Number 96865-92-8 Molecular Weight 428.48
Density 1.262g/cm3 Boiling Point N/A
Molecular Formula C21H28N6O4 Melting Point N/A
MSDS Chinese USA Flash Point N/A

 Use of Xanthine amine congener


Xanthine amine congener is a non-selective adenosine receptor antagonist[1]. Xanthine amine congener induces convulsions in mice[2].

 Names

Name N-(2-aminoethyl)-2-[4-(2,6-dioxo-1,3-dipropyl-7H-purin-8-yl)phenoxy]acetamide
Synonym More Synonyms

 Xanthine amine congener Biological Activity

Description Xanthine amine congener is a non-selective adenosine receptor antagonist[1]. Xanthine amine congener induces convulsions in mice[2].
Related Catalog
References

[1]. Ukena D, et al. Functionalized congeners of 1,3-dipropyl-8-phenylxanthine: potent antagonists for adenosine receptors that modulate membrane adenylate cyclase in pheochromocytoma cells, platelets and fat cells. Life Sci. 1986 Mar 3;38(9):797-807.

 Chemical & Physical Properties

Density 1.262g/cm3
Molecular Formula C21H28N6O4
Molecular Weight 428.48
Exact Mass 428.21700
PSA 137.03000
LogP 1.91820
Index of Refraction 1.586

 Safety Information

Personal Protective Equipment Eyeshields;Gloves;type N95 (US);type P1 (EN143) respirator filter
RIDADR NONH for all modes of transport
WGK Germany 3

 Articles30

More Articles
Chaperoning of the A1-adenosine receptor by endogenous adenosine - an extension of the retaliatory metabolite concept.

Mol. Pharmacol. 87(1) , 39-51, (2015)

Cell-permeable orthosteric ligands can assist folding of G protein-coupled receptors in the endoplasmic reticulum (ER); this pharmacochaperoning translates into increased cell surface levels of recept...

Allosteric interactions across native adenosine-A3 receptor homodimers: quantification using single-cell ligand-binding kinetics.

FASEB J. 25(10) , 3465-76, (2011)

A growing awareness indicates that many G-protein-coupled receptors (GPCRs) exist as homodimers, but the extent of the cooperativity across the dimer interface has been largely unexplored. Here, measu...

Hyperactivation of D1 and A2A receptors contributes to cognitive dysfunction in Huntington's disease.

Neurobiol. Dis. 74 , 41-57, (2015)

Stimulation of dopamine D1 receptor (D1R) and adenosine A2A receptor (A2AR) increases cAMP-dependent protein kinase (PKA) activity in the brain. In Huntington's disease, by essentially unknown mechani...

 Synonyms

Papaxac
XAC
Lopac-X-103
xanthine amine congener
Xanthine amine congener xac
Top Suppliers:I want be here



Get all suppliers and price by the below link:

Xanthine amine congener suppliers

Xanthine amine congener price