Teludipine-d6

Modify Date: 2024-01-09 19:15:38

Teludipine-d6 Structure
Teludipine-d6 structure
Common Name Teludipine-d6
CAS Number 1246833-02-2 Molecular Weight 504.65
Density N/A Boiling Point N/A
Molecular Formula C28H32D6N2O6 Melting Point N/A
MSDS N/A Flash Point N/A

 Use of Teludipine-d6


Teludipine-d6 (GR53992B-d6) is the deuterium labeled Teludipine hydrochloride. Teludipine is a lipophilic calcium channel blocker[1][2].

 Names

Name Teludipine-d6

 Teludipine-d6 Biological Activity

Description Teludipine-d6 (GR53992B-d6) is the deuterium labeled Teludipine hydrochloride. Teludipine is a lipophilic calcium channel blocker[1][2].
Related Catalog
In Vitro Stable heavy isotopes of hydrogen, carbon, and other elements have been incorporated into drug molecules, largely as tracers for quantitation during the drug development process. Deuteration has gained attention because of its potential to affect the pharmacokinetic and metabolic profiles of drugs[1].
References

[1]. Russak EM, et al. Impact of Deuterium Substitution on the Pharmacokinetics of Pharmaceuticals. Ann Pharmacother. 2019;53(2):211-216.

[2]. Tolomeo M, et al. Effects of R-enantiomer (GR66234A) and L-enantiomer (GR66235A) of telupidine, a new dihydropyridine derivative, on cell lines displaying the multidrug resistant phenotype. Haematologica. 1994 Jul-Aug;79(4):328-33.

 Chemical & Physical Properties

Molecular Formula C28H32D6N2O6
Molecular Weight 504.65