Name | BRL-44408 maleate |
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Synonyms |
BRL44408 maleate
2-[(4,5-dihydro-1H-imidazol-2-yl)methyl]-2,3-dihydro-1-methyl-1H-isoindole maleate 2-[(4,5-dihydro-1H-imidazol-2-yl)methyl]-2,3-dihydro-1-methyl-1H-isoindolemaleate 2-[(2H-1-methyl-1,3-dihydroisoindole)methyl]-4,5-dihydroimidazole maleate BRL 44408 maleate |
Description | BRL-44408 maleate is an α2A-adrenoceptor antagonist (Ki: 8.5 nM). BRL-44408 maleate has antidepressant and analgesic activity. BRL-44408 also improves cecal ligation puncture (CLP)-induced acute lung injury[1][2]. |
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Related Catalog | |
Target |
Ki: 8.5 nM (α2A-adrenoceptor)[1] |
References |
Molecular Formula | C17H21N3O4 |
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Molecular Weight | 331.36600 |
Exact Mass | 331.15300 |
PSA | 102.23000 |
LogP | 0.97900 |