2819989-60-9
2819989-60-9 structure
- Name: PBRM1-BD2-IN-4
- Chemical Name: PBRM1-BD2-IN-4
- CAS Number: 2819989-60-9
- Molecular Formula: C15H13ClN2O
- Molecular Weight: 272.73
- Catalog: Signaling Pathways Epigenetics Epigenetic Reader Domain
- Create Date: 2022-11-27 10:27:27
- Modify Date: 2024-04-05 17:16:11
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PBRM1-BD2-IN-4 (compound 15) is a potent PBRM1 Bromodomain inhibitor with Kd values of 5.5 μM and 11.1 μM for PBRM1-BD2 and PBRM1-BD5, respectively, and an IC50 value of 0.2 μM for PBRM1-BD2. PBRM1-BD2-IN-4 can be used to research anticancer[1].
| Name | PBRM1-BD2-IN-4 |
|---|
| Description | PBRM1-BD2-IN-4 (compound 15) is a potent PBRM1 Bromodomain inhibitor with Kd values of 5.5 μM and 11.1 μM for PBRM1-BD2 and PBRM1-BD5, respectively, and an IC50 value of 0.2 μM for PBRM1-BD2. PBRM1-BD2-IN-4 can be used to research anticancer[1]. |
|---|---|
| Related Catalog | |
| Target |
Kd: 5.5 μM (PBRM1-BD2), 11.1 μM (PBRM1-BD5)[1] IC50: 0.2 μM (PBRM1-BD2)[1] |
| Molecular Formula | C15H13ClN2O |
|---|---|
| Molecular Weight | 272.73 |