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  • DC Chemicals Limited
  • China
  • Product Name: PSB36
  • Price: $Inquiry/100mg $Inquiry/250mg $Inquiry/1g
  • Purity: 98.0%
  • Stocking Period: 3 Day
  • Contact: Tony Cao

524944-72-7

524944-72-7 structure
524944-72-7 structure
  • Name: PSB 36
  • Chemical Name: psb 36
  • CAS Number: 524944-72-7
  • Molecular Formula: C21H30N4O3
  • Molecular Weight: 386.48800
  • Create Date: 2017-07-12 01:55:43
  • Modify Date: 2024-01-02 12:39:33
  • PSB36 is a potent and selective antagonist of adenosine A1 receptor, with Kis 0.12 nM, 187 nM, 552 nM, 2300 nM, and 6500 nM for rA1, hA2B, rA2A, hA3 and rA3 receptors respectively. PSB36 can be used for the research of hyperalgesia[1][2].

Name psb 36
Synonyms hms3268h03
Description PSB36 is a potent and selective antagonist of adenosine A1 receptor, with Kis 0.12 nM, 187 nM, 552 nM, 2300 nM, and 6500 nM for rA1, hA2B, rA2A, hA3 and rA3 receptors respectively. PSB36 can be used for the research of hyperalgesia[1][2].
Related Catalog
Target

rA1:0.12 nM (Ki)

hA2B:187 nM (Ki)

rA2A:552 nM (Ki)

hA3:2300 nM (Ki)

rA3:6500 nM (Ki)

References

[1]. Abo-Salem OM, et, al. Antinociceptive effects of novel A2B adenosine receptor antagonists. J Pharmacol Exp Ther. 2004 Jan;308(1):358-66.

[2]. Bilkei-Gorzo A, et, al. Adenosine receptor subtype-selective antagonists in inflammation and hyperalgesia. Naunyn Schmiedebergs Arch Pharmacol. 2008 Mar;377(1):65-76.

Density 1.304g/cm3
Boiling Point 646.008ºC at 760 mmHg
Molecular Formula C21H30N4O3
Molecular Weight 386.48800
Flash Point 344.493ºC
Exact Mass 386.23200
PSA 92.91000
LogP 2.14650
Index of Refraction 1.616
RIDADR NONH for all modes of transport