GABAA receptor agent 5 structure
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Common Name | GABAA receptor agent 5 | ||
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CAS Number | 1808389-92-5 | Molecular Weight | 383.51 | |
Density | N/A | Boiling Point | N/A | |
Molecular Formula | C21H25N3O2S | Melting Point | N/A | |
MSDS | N/A | Flash Point | N/A |
Use of GABAA receptor agent 5GABAA receptor agent 5 (compound 018) is a potent γ-GABAAR antagonist with an Ki of 0.020 µM. GABAA receptor agent 5 shows γ-GABAAR antagonist activity with low cellular membrane permeability[1]. |
Name | GABAA receptor agent 5 |
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Description | GABAA receptor agent 5 (compound 018) is a potent γ-GABAAR antagonist with an Ki of 0.020 µM. GABAA receptor agent 5 shows γ-GABAAR antagonist activity with low cellular membrane permeability[1]. |
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Related Catalog | |
In Vitro | GABAA receptor agent 5 (compound 018) shows antagonist activity with IC50s of 0.24, 0.088, 0.068, 0.33, 0.79, 0.32, 0.079, 0.051 µM for α1β2δ, α4β1δ, α4β2δ, α6β2δ, α1β2γ2, α2β2γ2, α3β2γ2, α5β2γ2 subtypes, respectively[1]. |
References |
Molecular Formula | C21H25N3O2S |
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Molecular Weight | 383.51 |