(d(CH2)51,Tyr(Me)2,Arg8)-血管加压素

更新时间：2024-01-11 19:11:48

(d(CH2)51,Tyr(Me)2,Arg8)-血管加压素结构式	常用名	(d(CH2)51,Tyr(Me)2,Arg8)-血管加压素	英文名	(d(CH2)51,Tyr(Me)2,Arg8)-Vasopressin trifluoroacetate salt
	CAS号	73168-24-8	分子量	1151.36
	密度	1.5 g/cm3	沸点	N/A
	分子式	C₅₂H₇₄N₁₄O₁₂S₂	熔点	N/A
	MSDS	中文版美版	闪点	N/A
	符号	GHS07	信号词	Warning

(d(CH2)51,Tyr(Me)2,Arg8)-血管加压素用途

(d(CH2)51,Tyr(Me)2,Arg8)-Vasopressin (SKF 100273) 是一种vasopressin V1 受体选择性拮抗剂。

中文名	(D(CH2)51,TYR(ME)2,ARG8)-VASOPRESSIN
英文名	3-mercapto-3-methyl-butyryl-tyr(me)-phe-gln-asn-cys-pro-arg-gly-nh2
英文别名	更多

描述	(d(CH2)51,Tyr(Me)2,Arg8)-Vasopressin (SKF 100273) 是一种vasopressin V1 受体选择性拮抗剂。
相关类别	信号通路 >> G 蛋白偶联受体/G 蛋白 >> 血管加压素受体研究领域 >> 代谢疾病
参考文献	[1]. Arai Y, et al. New topics in vasopressin receptors and approach to novel drugs: research and development of conivaptan hydrochloride (YM087), a drug for the treatment of hyponatremia. J Pharmacol Sci. 2009 Jan;109(1):53-9.

密度	1.5 g/cm3
分子式	C₅₂H₇₄N₁₄O₁₂S₂
分子量	1151.36
精确质量	1150.51000
PSA	475.01000
LogP	3.52940
外观性状	白色冻干的粉末
折射率	1.695

符号	GHS07
信号词	Warning
危害声明	H332
个人防护装备	dust mask type N95 (US);Eyeshields;Gloves
危害码 (欧洲)	Xn: Harmful;
风险声明 (欧洲)	R20
安全声明 (欧洲)	36
危险品运输编码	NONH for all modes of transport

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In the current study, we aimed to determine the cardiovascular effects of arachidonic acid and peripheral mechanisms mediated these effects in normotensive conscious rats. Studies were performed in ma...

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Life Sci. 93(15) , 525-9, (2013)

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