![]() Ac-RYYRWK-NH2 TFA structure
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Common Name | Ac-RYYRWK-NH2 TFA | ||
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CAS Number | 408305-09-9 | Molecular Weight | 1126.19 | |
Density | N/A | Boiling Point | N/A | |
Molecular Formula | C51H70F3N15O11 | Melting Point | N/A | |
MSDS | N/A | Flash Point | N/A |
Use of Ac-RYYRWK-NH2 TFAAc-RYYRWK-NH2 is a potent and selective partial agonist for the nociceptin receptor (NOP), [3H]Ac-RYYRWK-NH2 binds to rat cortical membranes ORL1 with a Kd of 0.071 nM, but has no affinity for µ-, κ- or δ-opioid receptors[1]. |
Name | Ac-RYYRWK-NH2 TFA |
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Description | Ac-RYYRWK-NH2 is a potent and selective partial agonist for the nociceptin receptor (NOP), [3H]Ac-RYYRWK-NH2 binds to rat cortical membranes ORL1 with a Kd of 0.071 nM, but has no affinity for µ-, κ- or δ-opioid receptors[1]. |
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Related Catalog | |
In Vitro | [3H]ac-RYYRWK-NH2 binding to rat cortical membranes revealed a single high affinity site for [3H]ac-RYYRWK-NH2 (Kd=0.071 nM)[1]. Naloxone benzoylhydrazone displaced [3H]acRYYRWK-NH2 binding to rat cortical membranes (Ki=104 nM) and human ORL1 (Ki=136 nM) as well as [125I]Tyr14-NC-OH to ORL1 (Ki=37 nM) has no affinity for µ-, κ- or δ-opioid receptors[1]. |
References |
Molecular Formula | C51H70F3N15O11 |
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Molecular Weight | 1126.19 |