Glutathione-S-transferases (GSTs) are a family of Phase II detoxification enzymes that catalyse the conjugation of glutathione (GSH) to a wide variety of endogenous and exogenous electrophilic compounds. GSTs are divided into two distinct super-family members: the membrane-bound microsomal and cytosolic family members. Microsomal GSTs are structurally distinct from the cytosolic in that they homo- and heterotrimerize rather than dimerize to form a single active site. Microsomal GSTs play a key role in the endogenous metabolism of leukotrienes and prostaglandins. Glutathione S-transferases (GSTs) function to protect cellular macromolecules from attack by reactive electrophiles. GSTs may be viable drug targets in disease states unrelated to cancer.


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GSTO-IN-2

GSTO-IN-2 is a glutathione S-transferase inhibitor with IC50s of 3.6, 16.3, and 1.4 μM for GSTA2, GSTM1, and GSTP1-1.

  • CAS Number: 1202710-57-3
  • MF: C33H52N2O9
  • MW: 620.77
  • Catalog: Gutathione S-transferase
  • Density: N/A
  • Boiling Point: N/A
  • Melting Point: N/A
  • Flash Point: N/A

AZD9898

AZD9898 is an orally active leukotriene-C4 synthetase (LTC4S, glutathione S-transferase II) inhibitor, with an IC50 of 0.28 nM. AZD9898 mitigates the GABA binding and hepatic toxicity signal. AZD9898 has the potential to treat asthma[1].

  • CAS Number: 2042347-69-1
  • MF: C20H19ClF3N3O4
  • MW: 457.83
  • Catalog: Gutathione S-transferase
  • Density: N/A
  • Boiling Point: N/A
  • Melting Point: N/A
  • Flash Point: N/A

GSTO1-IN-1

GSTO1-IN-1 is a potent glutathione S-transferase omega 1 (GSTO1) inhibitor with an IC50 of 31 nM.

  • CAS Number: 568544-03-6
  • MF: C10H12Cl2N2O3S
  • MW: 311.185
  • Catalog: Gutathione S-transferase
  • Density: 1.5±0.1 g/cm3
  • Boiling Point: N/A
  • Melting Point: N/A
  • Flash Point: N/A

ezatiostat

Ezatiostat is a glutathione analog inhibitor of glutathione S-transferase P1-1 (GSTP1-1).

  • CAS Number: 168682-53-9
  • MF: C27H35N3O6S
  • MW: 529.648
  • Catalog: Gutathione S-transferase
  • Density: 1.2±0.1 g/cm3
  • Boiling Point: 749.7±60.0 °C at 760 mmHg
  • Melting Point: N/A
  • Flash Point: 407.2±32.9 °C

Curzerene

Curzerene is a sesquiterpene is isolated from the rhizome of Curculigo orchioides Gaertn with anti-cancer activity. Curzerene inhibits glutathione S-transferase A1 (GSTA1) mRNA and protein expression. Curzerene induces cell apoptosis[1].

  • CAS Number: 17910-09-7
  • MF: C15H20O
  • MW: 216.319
  • Catalog: Gutathione S-transferase
  • Density: 1.0±0.1 g/cm3
  • Boiling Point: 282.8±40.0 °C at 760 mmHg
  • Melting Point: N/A
  • Flash Point: 117.5±14.2 °C

Alpha-Angelica lactone

α-Angelica lactone is a naturally occurring anticarcinogen and an vinylogous nucleophile. α-Angelica lactone can give the chiral δ-amino γ,γ-disubstituted butenolide carbonyl derivatives and exhibitselectrophilic trapping at the γ-carbon. α-Angelica lactone exerts strong chemoprotective effects by selective enhancement of glutathione-S-thansferase (GST) and UDP-glucononosyltransferase (UGT) detoxification enzymes[1][2][3][4].

  • CAS Number: 591-12-8
  • MF: C5H6O2
  • MW: 98.100
  • Catalog: Gutathione S-transferase
  • Density: 1.1±0.1 g/cm3
  • Boiling Point: 249.4±9.0 °C at 760 mmHg
  • Melting Point: 13-17 °C(lit.)
  • Flash Point: 68.3±0.0 °C

Sperabillin A dihydrochloride

Sperabillin A (dihydrochloride)is new inhibitors ofglutathione S-transferaseisolated from the culture broth ofStreptomyces sp[1].

  • CAS Number: 111337-87-2
  • MF: C15H29Cl2N5O3
  • MW: 398.32800
  • Catalog: Gutathione S-transferase
  • Density: N/A
  • Boiling Point: N/A
  • Melting Point: N/A
  • Flash Point: N/A

Ethacrynic acid D5

Ethacrynic acid D5 is a deuterium labeled Ethacrynic acid. Ethacrynic acid is a diuretic. Ethacrynic acid is an inhibitor of glutathione S-transferases (GSTs). Ethacrynic acid is a potent inhibitor of NF-kB-signaling pathway, and also modulates leukotriene formation. Ethacrynic acid also inhibits L-type voltage-dependent and store-operated calcium channel, leading to relaxation of airway smooth muscle (ASM) cells. Ethacrynic acid has anti-inflammatory properties that reduces the retinoid-induced ear edema in mice[1][2][3][4].

  • CAS Number: 1330052-59-9
  • MF: C13H7D5Cl2O4
  • MW: 308.169
  • Catalog: Calcium Channel
  • Density: 1.4±0.1 g/cm3
  • Boiling Point: 480.0±45.0 °C at 760 mmHg
  • Melting Point: N/A
  • Flash Point: 244.1±28.7 °C

(-)-Anonaine

Anonaine is an antiparasitic agent. Anonaine also is a glutathione S-transferase (GST) inhibitor[1].

  • CAS Number: 1862-41-5
  • MF: C17H15NO2
  • MW: 265.31
  • Catalog: Gutathione S-transferase
  • Density: 1.294g/cm3
  • Boiling Point: 444.7ºC at 760mmHg
  • Melting Point: N/A
  • Flash Point: 177.1ºC

Ethacrynic acid

Ethacrynic acid is a diuretic. Ethacrynic acid is an inhibitor of glutathione S-transferases (GSTs). Ethacrynic acid is a potent inhibitor of NF-kB-signaling pathway, and also modulates leukotriene formation. Ethacrynic acid also inhibits L-type voltage-dependent and store-operated calcium channel, leading to relaxation of airway smooth muscle (ASM) cells. Ethacrynic acid has anti-inflammatory properties that reduces the retinoid-induced ear edema in mice[1][2][3][4].

  • CAS Number: 58-54-8
  • MF: C13H12Cl2O4
  • MW: 303.13800
  • Catalog: Calcium Channel
  • Density: 1.35g/cm3
  • Boiling Point: 480ºC at 760mmHg
  • Melting Point: 125 °C
  • Flash Point: 244.1ºC

Coniferyl ferulate

Coniferyl ferulate, a strong inhibitor of glutathione S-transferase (GST) isolated from Radix Angelicae sinensis, reverses multidrug resistance and downregulates P-glycoprotein. Coniferyl ferulate shows strong inhibition of human placental GST with an IC50 of 0.3 μM[1].

  • CAS Number: 63644-62-2
  • MF: C20H20O6
  • MW: 356.369
  • Catalog: P-glycoprotein
  • Density: 1.3±0.1 g/cm3
  • Boiling Point: 570.5±50.0 °C at 760 mmHg
  • Melting Point: N/A
  • Flash Point: 202.8±23.6 °C

Seneciphylline

Seneciphylline is a toxic pyrrolizidine alkaloid in Senecio plants[1]. Seneciphylline significantly increases the activities of epoxide hydrase and glutathione-S-transferase but causes reduction of cytochrome P-450 and related monooxygenase activities[2].

  • CAS Number: 480-81-9
  • MF: C18H23NO5
  • MW: 333.379
  • Catalog: Cytochrome P450
  • Density: 1.3±0.1 g/cm3
  • Boiling Point: 577.7±50.0 °C at 760 mmHg
  • Melting Point: 217ºC
  • Flash Point: 303.2±30.1 °C

Ezatiostat (hydrochloride)

Ezatiostat hydrochloride is a glutathione analog inhibitor of glutathione S-transferase P1-1 (GSTP1-1).

  • CAS Number: 286942-97-0
  • MF: C27H36ClN3O6S
  • MW: 566.109
  • Catalog: Gutathione S-transferase
  • Density: N/A
  • Boiling Point: N/A
  • Melting Point: N/A
  • Flash Point: N/A

TLK117

TLK117, the active metabolite of TLK199, selective inhibits Glutathione S-transferase P1–1 (GSTP1-1) with a Ki of 0.4 μM for GSTP. TLK117 also competitively inhibits glyoxalase I with a Ki of 0.56 μM.

  • CAS Number: 152684-53-2
  • MF: C23H27N3O6S
  • MW: 473.54
  • Catalog: Gutathione S-transferase
  • Density: N/A
  • Boiling Point: N/A
  • Melting Point: N/A
  • Flash Point: N/A

TK05

TK05 is a potent and selective inhibitor of leukotriene C4 synthase (LTC4S) with an IC50 of 95 nM[1].

  • CAS Number: 1245734-61-5
  • MF: C31H25ClN2O5
  • MW: 540.99
  • Catalog: Gutathione S-transferase
  • Density: N/A
  • Boiling Point: N/A
  • Melting Point: N/A
  • Flash Point: N/A

LAS17

Novel highly potent, selective, and irreversible GSTP1 inhibitor

  • CAS Number: 2362527-67-9
  • MF: C15H20Cl2N4O2
  • MW: 359.25
  • Catalog: Gutathione S-transferase
  • Density: N/A
  • Boiling Point: N/A
  • Melting Point: N/A
  • Flash Point: N/A

BRD2889

BRD2889 is an analog of the alkaloid piperlongumine. BRD2889 is a robust modulator of the GSTP1-ISCU axis in pulmonary hypertension (PH)[1].

  • CAS Number: 1415153-39-7
  • MF: C26H25NO6
  • MW: 447.48
  • Catalog: Gutathione S-transferase
  • Density: N/A
  • Boiling Point: N/A
  • Melting Point: N/A
  • Flash Point: N/A

7-Acetoxy-4-methylcoumarin

7-Acetoxy-4-methylcoumarin is an inhibitor of GST.7-Acetoxy-4-methylcoumarin inhibits AFB1-DNA binding in vitro with 36.7% inhibition[1][2].

  • CAS Number: 2747-05-9
  • MF: C12H10O4
  • MW: 218.20500
  • Catalog: Gutathione S-transferase
  • Density: 1.263g/cm3
  • Boiling Point: 371.4ºC at 760mmHg
  • Melting Point: 149-150 °C(lit.)
  • Flash Point: 191.5ºC

Ethacrynic acid sodium

Ethacrynic acid (Etacrynic acid sodium) sodium is a diuretic. Ethacrynic acid sodium is an inhibitor of glutathione S-transferases (GSTs). Ethacrynic acid sodium is a potent inhibitor of NF-kB-signaling pathway, and also modulates leukotriene formation. Ethacrynic acid sodium also inhibits L-type voltage-dependent and store-operated calcium channel, leading to relaxation of airway smooth muscle (ASM) cells. Ethacrynic acid sodium has anti-inflammatory properties that reduces the retinoid-induced ear edema in mice[1][2][3][4].

  • CAS Number: 6500-81-8
  • MF: C13H11Cl2NaO4
  • MW: 325.12
  • Catalog: Calcium Channel
  • Density: N/A
  • Boiling Point: 480ºC at 760 mmHg
  • Melting Point: 121-122ºC
  • Flash Point: 244.1ºC